• Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
  • Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
  • Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
  • Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
  • Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
  • Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib

Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib

Powder: Yes
Customized: Customized
Certification: GMP, HSE, ISO 9001, USP, BP
Suitable for: Elderly, Adult
State: Powder
Purity: >99%
Samples:
US$ 120/g 1 g(Min.Order)
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Customization:
Diamond Member Since 2021

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  • Overview
  • Product Description
  • Product Details
  • Application&Function
  • Specification
Overview

Basic Info.

Model NO.
D-sung Ponatinib
Product Name
Ponatinib
Name
Ponatinib Powder
Appearance
Yellow Powder
Color
Yellow
Grade
Pharmaceutical Grade
Assay
HPLC 99%
Application
Pharmaceutical
Specific
COA
Test Method
HPLC
Shelf Life
2 Years
CAS No.
943319-70-8
Mf
C29h27f3n6o
MW
532.56
Melting Point
>175 C
Density
1.292
Transport Package
Negotiable
Specification
99%
Trademark
D-sung
Origin
Shaanxi Xi′an
Production Capacity
1000kg/Month

Product Description

Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
Product Description
Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder PonatinibPharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
Product Details
Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
 
Product Name Ponatinib
Appearance Yellow Powder
CAS No. 943319-70-8
MF C29H27F3N6O

Ponatinib is an anticancer drug. It was approved by FDA in December 2012 for the treatment of adult chronic myelogenous leukemia (CML) and "Philadelphia chromosome positive" (PH +) acute lymphoblastic leukemia (ALL). It is mainly used to treat patients who do not respond to dasatinib or nillotinib therapy, or who are unable to tolerate dasatinib or nillotinib, and who are not suitable for subsequent treatment with imatinib. It can also be used to treat patients with a genetic mutation (the "T315I mutation") that makes patients resistant to imatinib, dasatinib, or nilotinib. It is also used to treat CML and pH +ALL in adults who have not been treated with other TKIs. It is currently the only marketed drug that is effective against the BCR-ABL kinase T315I mutation. 

Application&Function
Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib

Ponatinib was approved in the European Union in July 2013 through a centralised approval process. Panatinib is the third generation of multi-target tyrosine kinase inhibitors. Typical drugs of multi-target tyrosine kinase inhibitors include sunitinib, imatinib, sorafenib and vataranib., for he (Ponatinib) can effectively inhibit the in vitro FGFR1-4 kinase activity, its IC50 alue concentration,2,18 2 and 8 nmol/L respectively, in the absence of interleukin - 3 cells, FGFR1, on behalf of, to curb cells - 4 kinase expression of IC50 alue concentration were 8 August 24 and 34 nmol/L, and tested in each cell, for inhibition of FGFR1-4 phosphorylation, its IC50 alue concentration is 39 29 32 and 39 nmol/L respectively tested on endometrial bladder Stomach and thymus in multiple cell lines FGFR inhibition, relatively, compared with other drugs for showed obvious pharmacological effects, such as its inhibit endometrial AN3CA and MFE - 296 cell proliferation GI50 value of 14 and 61 nmol/L, it shows that, for he is a powerful FGFR inhibitors in mice tumor xenograft model, each day 10 mg/kg or 30 mg/kg, tumor inhibition rate were 49% and 82%, respectively.

Specification
Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder PonatinibPharmaceutical Grade Ponatinib Raw Material Ponatinib Powder PonatinibPharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder PonatinibPharmaceutical Grade Ponatinib Raw Material Ponatinib Powder PonatinibPharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
Pharmaceutical Grade Ponatinib Raw Material Ponatinib Powder Ponatinib
 

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Diamond Member Since 2021

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Management System Certification
ISO 9001, ISO 14001, GMP, HACCP