Anti-Anxiety Tianeptine Sodium Powder Nootropics Tianeptine Sodium
Product Description
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Product Details
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Product Name |
Tianeptine Sodium |
Appearance |
White Powder |
CAS |
30123-17-2 |
Molecular Formu |
C21h24cln2nao4s |
Density |
1.38 |
Tinepin sodium salt is a tricyclic antidepressant drug, and its antidepressant mechanism is different from traditional tricyclic antidepressants. It can increase the reuptake of 5-HT in synaptic cleft and may have an effect on improving 5-HT neuronal conduction. Has no affinity for cholinergic or adrenergic receptors. The antidepressant efficacy is similar to tricyclic drugs, but the tolerability is better than tricyclic drugs. In animal experiments, it can increase the spontaneous activity of pyramidal cells in the hippocampus and accelerate their recovery after functional inhibition; Can increase the reabsorption of serotonin by neurons in the cerebral cortex and hippocampus.
Thiamethasone sodium is rapidly and completely absorbed in the digestive tract. The distribution is rapid, with a PPB of up to 94%. In the liver, complete metabolism is achieved through β - oxidation and N-demethylation, and the clearance of terminal T1/2 is short, taking 2.5 hours. A very small amount of the original drug (8%) is excreted from the kidneys, mainly its metabolites are excreted from the urine. The clearance of T1/2 in patients with renal insufficiency is prolonged by 1 hour.
Application&Function
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Sodium salt of tianeptin, also known as tianeptin sodium; Datilang; Sulfamethoxazole; Thionaproxen is a novel tricyclic antidepressant that exerts antidepressant effects by acting on the 5-HT system. It is mainly used clinically to treat mild, moderate, or severe depression, neurogenic and reactive depression, anxiety and depression caused by physical discomfort, especially gastrointestinal discomfort, and anxiety and depression in alcohol dependent patients during withdrawal.
Tinepin sodium salt has a good effect on mood disorders and physical discomfort symptoms.
The combination of tianeptin sodium and monoamine oxidase inhibitors can cause cardiovascular disease attacks or paroxysmal hypertension, high fever, convulsions, and even death. Before taking this product, the monoamine oxidase inhibitor must be discontinued for 2 weeks. After discontinuing this product for 24 hours, monoamine oxidase inhibitors can be taken.
Salicylic acid salts can reduce the plasma protein binding rate of this product, and should be reduced when used in combination.